We are cultivating a differentiated pipeline of small molecule medicines that utilize first-in-class or potential best-in-class mechanisms of action (MoAs) to restore balance in the brain by reducing the neuronal hyperexcitability that underlies debilitating brain conditions. Our unique understanding of the complexities of neurologic systems allows us to turn preclinical potential into clinical results.

Our aim is to make a meaningful impact and address the significant unmet need in the lives of individuals with neurological disorders that present with brain conditions.

Publications and Posters ยป

Programs Indication opportunities Preclinical Phase 1 Phase 2
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OV329, a next-generation GABA-aminotransferase inhibitor
GABA-aminotransferase inhibitor Drug resistant adult focal onset seizures (FOS)
Tuberous sclerosis complex seizures (TSC)
Infantile spasms (IS)
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OV4071, Potassium-chloride cotransporter 2 (KCC2) direct activator (oral)
OV4071 Psychosis assoc. with Parkinson's disease and Lewy body dementia and acute schizophrenia

Ketamine challenge with biomarkers

Program/Indication Stage
OV329, a next-generation GABA-aminotransferase inhibitor

GABA-aminotransferase inhibitor Drug resistant adult focal onset seizures (FOS)

Phase 2

GABA-aminotransferase inhibitor Drug resistant adult focal onset seizures (FOS)

Phase 2

GABA-aminotransferase inhibitor Tuberous sclerosis complex seizures (TSC)

Phase 2

GABA-aminotransferase inhibitor Infantile spasms (IS)

Phase 2

Program/Indication Stage
OV4071, Potassium-chloride cotransporter 2 (KCC2) direct activator (oral)

OV4071 Psychosis assoc. with Parkinson's disease and Lewy body dementia and acute schizophrenia

Phase 1

OV4071 Psychosis assoc. with Parkinson's disease and Lewy body dementia and acute schizophrenia
Ketamine challenge with biomarkers

Phase 1

*Timelines pending feedback from regulatory discussions Ketamine challenge to initiate pending PK characterization in Phase 1 study